SCHEMBL7285015

SCHEMBL7285015

CC(C)(C)OC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ccc(C#N)nc3)cc2)NC1=O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
GPR119 Q8TDV5 3/20 0.43
IRAK4 Q9NWZ3 2/20 0.35
CTSC P53634 2/20 0.35
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
KCNH2 Q12809 2/20 0.33
TRPA1 O75762 1/20 0.33
JAK2 O60674 1/20 0.33
BRD4 O60885 1/20 0.33
CHEK1 O14757 1/20 0.32
DPP4 P27487 2/20 0.32
VHL P40337 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285264 0.89 ITGB3 (0.53) ITGB3ITGA2BGPR119BRD4DPP4
SCHEMBL7277677 0.89 ITGB3 (0.46) ITGB3ITGA2BGPR119IRAK4CTSC
SCHEMBL8884076 0.89 ITGB3 (0.52) ITGB3ITGA2BGPR119BRD4DPP4
SCHEMBL7283463 0.87 ITGB3 (0.49) ITGB3ITGA2BGPR119IRAK4BRD4
SCHEMBL7275877 0.85 ITGB3 (0.46) ITGB3ITGA2BGPR119IRAK4CTSC
Hydrochloric Acid SCHEMBL7275160 0.84 ITGB3 (0.58) ITGB3ITGA2BGPR119IRAK4
SCHEMBL7286097 0.84 ITGB3 (0.44) ITGB3ITGA2BGPR119IRAK4BRD4
Hydrochloric Acid SCHEMBL7275246 0.83 ITGB3 (0.58) ITGB3ITGA2BGPR119IRAK4
SCHEMBL7323680 0.83 ITGB3 (0.47) ITGB3ITGA2BGPR119CTSCTRPA1
SCHEMBL7318086 0.83 ITGB3 (0.47) ITGB3ITGA2BIRAK4CTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed