SCHEMBL7277556

SCHEMBL7277556

CC(C)(C)OC(=O)CC[CH]Oc1cccc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 3/20 0.49
HSD17B10 Q99714 2/20 0.49
HPGD P15428 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
PGR P06401 1/20 0.40
GAA P10253 1/20 0.40
PTGS1 P23219 1/20 0.40
MAPK1 P28482 1/20 0.40
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NR1D1 P20393 2/20 0.39
OGG1 O15527 1/20 0.38
BTN3A1 O00481 3/20 0.38
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6707308 0.83 TNF (0.46) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL9439620 0.80 ALDH1A1 (0.55) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL7279601 0.79 ALDH1A1 (0.46) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL7277563 0.78 CNR2 (0.54) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL6708188 0.78 MRGPRX4 (0.45) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL5161970 0.76 ALDH1A1 (0.62) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL7278827 0.75 ALDH1A1 (0.51) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL6707441 0.75 ALDH1A1 (0.45) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL6446932 0.75 ALDH1A1 (0.42) ALDH1A1KDM4EHSD17B10HPGDTDP1
SCHEMBL6447173 0.74 ALDH1A1 (0.44) ALDH1A1KDM4EHSD17B10HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5278148-A Hypotensive agents HOFFMANN-LA ROCHE INC. (US) 1994-01-11 US disclosed
US-5140011-A Hypotensive agents HOFFMANN-LA ROCHE, INC. (US) 1992-08-18 US disclosed
EP-0391179-A2 Peptide derivatives of amino acids having a renin-inhibiting effect F. HOFFMANN-LA ROCHE AG (CH) 1990-10-10 EP disclosed
EP-0391180-A2 Peptide derivatives of amino acids having a renin-inhibiting effect F. HOFFMANN-LA ROCHE AG (CH) 1990-10-10 EP disclosed
EP-0389898-A2 Peptide derivatives of amino acids having a renin-inhibiting effect F. HOFFMANN-LA ROCHE AG (CH) 1990-10-03 EP disclosed
US-4931591-A Novel 5-amino-4-hydroxyvaleryl derivatives CIBA-GEIGY CORPORATION (US) 1990-06-05 US disclosed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US disclosed
EP-0184550-A2 5-Amino-4-hydroxy valeryl amide derivatives CIBA-GEIGY AG (CH) 1986-06-11 EP disclosed