SCHEMBL7278250

SCHEMBL7278250

COC(=O)CCN1C(=O)COc2ccc(C(N)C(=O)OC(C)(C)C)cc21

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
KMO O15229 1/20 0.44
CYP3A4 P08684 4/20 0.43
CYP2C19 P33261 4/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 2/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
HTT P42858 1/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2D6 P10635 2/20 0.42
POLB P06746 4/20 0.41
HSD17B10 Q99714 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270151 0.90 KMO (0.56) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL7270859 0.81 POLB (0.41) TSHRALDH1A1USP2POLBTP53
SCHEMBL7278244 0.78 CYP3A4 (0.54) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL16897914 0.77 TSHR (0.69) TSHRCYP3A4CYP2C19ALDH1A1CYP1A2
SCHEMBL7268703 0.74 KMO (0.51) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL31444652 0.72 TSHR (0.46) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL18264378 0.71 KMO (0.50) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL7278012 0.71 ALDH1A1 (0.38) TSHRCYP2C19ALDH1A1USP2CYP2C9
SCHEMBL5799939 0.71 KMT2A (0.47) TSHRKMOCYP3A4CYP2C19ALDH1A1
SCHEMBL7270138 0.69 KMO (0.56) TSHRKMOCYP3A4CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445467-A1 Renin inhibitors and antiviral agents Beecham Group p.l.c. (GB) 1991-09-11 EP disclosed
EP-0411751-A1 Renin inhibitory peptides Beecham Group p.l.c. (GB) 1991-02-06 EP disclosed