SCHEMBL7278536

SCHEMBL7278536

CCc1noc(CNC=O)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALOX15 P16050 1/20 0.35
APOBEC3A P31941 1/20 0.35
HSD17B10 Q99714 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADH1B P00325 1/20 0.30
ADH1A P07327 1/20 0.30
ADH7 P40394 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7288646 0.86 APOBEC3A (0.43) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL7279260 0.81 ROCK2 (0.37) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL7291657 0.78 MAPT (0.41) HSD17B10ADH1BADH1AADH7MAPT
SCHEMBL9966023 0.77 L3MBTL1 (0.35) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL8882150 0.75 NPC1 (0.36) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL7291628 0.75 KDM4E (0.35) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL12705 0.74
SCHEMBL7392164 0.73 L3MBTL1 (0.36) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL9963365 0.73 KDM4E (0.33) KDM4EALOX15APOBEC3AHSD17B10APOBEC3G
SCHEMBL3307623 0.70 ADH1B (0.31) ADH1BADH1AADH7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0320136-B1 Imidazoquinoxaline compounds and their preparation and use NOVO NORDISK AS (DK) 1994-07-27 EP disclosed
EP-0311321-B1 Heterocyclic compounds and their preparation and use NOVO NORDISK AS (DK) 1994-01-12 EP disclosed
EP-0283162-B1 HETEROCYCLIC COMPOUNDS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1993-08-11 EP disclosed
EP-0274009-B1 OXADIAZOLYLACETONITRILES, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-09-09 EP disclosed
US-4999354-A Central Nervous System Disorders, Anticonvulsant and Anxiolytic Agents A/S FERROSAN (DK) 1991-03-12 US disclosed
EP-0241682-B1 NOVEL BENZODIAZEPINE DERIVATIVES AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1990-11-28 EP disclosed
US-4968682-A CENTRAL NERVOUS SYSTEM DISORDERS A/S FERROSAN (DK) 1990-11-06 US disclosed
US-4902686-A Tricyclic heterocyclic compounds and their use in treating benzodiazepin receptor-related ailments A/S FERROSAN (DK) 1990-02-20 US disclosed
US-4886797-A CENTRAL NERVOUS SYSTEM DISORDERS A/S FERROSAN (DK) 1989-12-12 US disclosed
US-4880799-A CENTRAL NERVOUS SYSTEM DISORDERS, ANTICONVULSANTS A/S FERROSAN (DK) 1989-11-14 US disclosed
EP-0283162-A2 Heterocyclic compounds and their preparation and use NOVO NORDISK A/S (DK) 1988-09-21 EP disclosed
US-4772599-A ANTICONVULSANTS, ANXIOLYTICS, HYPNOTICS, NOOTROPICS A/S FERROSAN (DK) 1988-09-20 US disclosed
US-4771051-A CENTRAL NERVOUS SYSTEM DISORDERS A/S FERROSAN (DK) 1988-09-13 US disclosed
US-4727153-A NERVOUS SYSTEM DISORDERS A/S FERROSAN (DK) 1988-02-23 US disclosed
EP-0241682-A2 Novel benzodiazepine derivatives and their preparation and use NOVO NORDISK A/S (DK) 1987-10-21 EP disclosed
EP-0226282-A2 Heterocyclic compounds and their preparation and use A/S FERROSAN (DK) 1987-06-24 EP disclosed
EP-0225013-A1 Heterocyclic compounds and their preparation and use A/S FERROSAN (DK) 1987-06-10 EP disclosed
US-4670433-A CARDIOVASCULAR DISORDERS A/S FERROSAN (DK) 1987-06-02 US disclosed
EP-0220845-A1 Heterocyclic compounds and their preparation and use A/S FERROSAN (DK) 1987-05-06 EP disclosed
EP-0197282-A1 Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds A/S FERROSAN (DK) 1986-10-15 EP disclosed