SCHEMBL7278918

SCHEMBL7278918

CN1C(=O)COc2c(C(=O)O)cc([N+](=O)[O-])cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 2/20 0.40
TDP1 Q9NUW8 3/20 0.39
HTR2A P28223 1/20 0.39
SLC6A4 P31645 1/20 0.39
HRH1 P35367 1/20 0.39
HTR3A P46098 1/20 0.39
PDE4D Q08499 1/20 0.39
KCNH2 Q12809 1/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 2/20 0.38
MAPK1 P28482 1/20 0.38
GAA P10253 2/20 0.38
TP53 P04637 1/20 0.36
LMNA P02545 2/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7290643 0.99 ALDH1A1 (0.40) ALDH1A1SMN1; SMN2HTTTDP1HTR2A
SCHEMBL7290637 0.89 HTR2A (0.41) ALDH1A1SMN1; SMN2HTTTDP1HTR2A
SCHEMBL20265127 0.80 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2HTTTDP1HTR2A
SCHEMBL7287945 0.80 PDE3B (0.49) ALDH1A1HTTTDP1HTR2ASLC6A4
SCHEMBL7288619 0.79 PDE4D (0.57) HTTTDP1HTR2ASLC6A4HRH1
Hydrochloric Acid SCHEMBL7291531 0.79 PDE3B (0.48) ALDH1A1HTTTDP1HTR2ASLC6A4
SCHEMBL7269116 0.78 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2HTTCYP1A2MAPT
Hydrochloric Acid SCHEMBL7290566 0.77 PDE4D (0.56) HTTTDP1HTR2ASLC6A4HRH1
SCHEMBL7291597 0.76 HTR3A (0.73) ALDH1A1SMN1; SMN2TDP1HTR2ASLC6A4
SCHEMBL7290641 0.76 HTT (0.39) ALDH1A1SMN1; SMN2HTTTDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0313393-B1 Benzoxazine compounds and pharmaceutical use thereof YOSHITOMI PHARMACEUTICAL (JP) 1994-03-16 EP disclosed
US-4892872-A ANTIEMETICS, ANTINAUSEA YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed
EP-0313393-A2 Benzoxazine compounds and pharmaceutical use thereof Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-04-26 EP disclosed