SCHEMBL7279397

SCHEMBL7279397

CO[C@H]1C(=O)N2C(C(=O)OC(C)(C)C)=C(C)CS(=O)(=O)C12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7970632 1.00 ELANE (1.00) ELANE
SCHEMBL7436377 1.00 ELANE (1.00) ELANE
SCHEMBL7436386 1.00 ELANE (1.00) ELANE
SCHEMBL7432470 0.86 ELANE (0.76) ELANE
SCHEMBL7432478 0.86 ELANE (0.76) ELANE
SCHEMBL7271778 0.86 ELANE (0.76) ELANE
SCHEMBL8399288 0.85 ELANE (1.00) ELANE
SCHEMBL8399285 0.85 ELANE (1.00) ELANE
SCHEMBL8670544 0.84 ELANE (0.72) ELANE
SCHEMBL8670547 0.84 ELANE (0.72) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5364848-A Elastase inhibitors MERCK & CO., INC. (US) 1994-11-15 US disclosed
US-5356888-A Elastase inhibitors FARMITALIA CARLO ERBA (IT) 1994-10-18 US disclosed
EP-0378604-B1 1,1-DIOXO-CEPHEM-4-CARBOTHIOLIC ACID DERIVATIVES ERBA CARLO SPA (IT) 1994-03-02 EP disclosed
US-5132301-A Substituted cephalosporin sulfones as anti-inflammatory and anti-degenerative agents MERCK & CO., INC. (US) 1992-07-21 US disclosed
EP-0378604-A1 1,1-DIOXO-CEPHEM-4-CARBOTHIOLIC ACID DERIVATIVES. ERBA CARLO SPA (IT) 1990-07-25 EP disclosed
WO-1989010926-A1 1,1-DIOXO-CEPHEM-4-CARBOTHIOLIC ACID DERIVATIVES FARMITALIA CARLO ERBA S.R.L. (IT) 1989-11-16 WO disclosed
EP-0267723-A2 New substituted cephalosporin sulfones as anti-inflammatory and anti-degenerative agents MERCK & CO. INC. (US) 1988-05-18 EP disclosed
EP-0124081-A2 New substituted cephalosporin sulfones as antiinflammatory and antidegenerative agents, pharmaceutical compositions containing the same and processes for making them MERCK & CO. INC. (US) 1984-11-07 EP disclosed