SCHEMBL7279472

SCHEMBL7279472

COc1ccc(CCN(CCc2ccccc2)C(=O)C2CCC(C(N)=O)CC2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
LPAR1 Q92633 2/20 0.50
LPAR5 Q9H1C0 2/20 0.50
CHRM5 P08912 2/20 0.50
CHRM1 P11229 2/20 0.50
CHRM3 P20309 2/20 0.50
HTR2A P28223 2/20 0.49
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49
PLAAT3 P53816 1/20 0.49
PLAAT5 Q96KN8 1/20 0.49
PLAAT2 Q9NWW9 1/20 0.49
PLAAT4 Q9UL19 1/20 0.49
ALDH1A1 P00352 1/20 0.48
ADRB1 P08588 1/20 0.48
HTR1A P08908 1/20 0.48
ADRA2A P08913 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993505 0.75 L3MBTL1 (0.58) L3MBTL1HTR2AHTR2CHTR2BPLAAT3
SCHEMBL7279469 0.75 ALDH1A1 (0.71) KDM4ENPC1RAB9APLAAT3PLAAT5
SCHEMBL8098593 0.75 L3MBTL1 (0.58) L3MBTL1LPAR1HTR2AHTR2CHTR2B
SCHEMBL7279475 0.75 ALDH1A1 (0.71) KDM4ENPC1RAB9APLAAT3PLAAT5
SCHEMBL28901341 0.74 L3MBTL1 (0.57) KDM4EL3MBTL1HTR2AHTR2CHTR2B
Methylamine SCHEMBL10385050 0.72 CYP19A1 (0.71) KDM4E
SCHEMBL12971411 0.72 EBP (0.68) KDM4EPLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL10526510 0.72 EBP (0.68) KDM4EPLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL8604705 0.72 CYP19A1 (0.70) KDM4EALDH1A1
SCHEMBL30173445 0.72 CYP19A1 (0.70) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375668-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1990-06-27 EP disclosed
US-4885313-A 3,4-Dihydroxyphenylethylamine derivatives and their use FISONS PLC (GB) 1989-12-05 US disclosed
US-4803225-A Dihydroxy-phenethylamino compounds useful as pharmaceuticals FISONS, PLC (GB) 1989-02-07 US disclosed
US-4720586-A Substituted 3,4-dihydroxy-phenylethylamino compounds FISONS, PLC (GB) 1988-01-19 US disclosed
EP-0142283-A2 Phenylethylamines, process for their preparation and compositions containing them FISONS plc (GB) 1985-05-22 EP disclosed