SCHEMBL7280200

SCHEMBL7280200

CCOC(=O)OC1(CNCc2ccc(-c3ccccc3C#N)cc2)CCCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.44
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
MYC P01106 1/20 0.42
WDR5 P61964 1/20 0.42
FFAR1 O14842 1/20 0.38
AKR1B1 P15121 1/20 0.38
ADAM17 P78536 1/20 0.38
MME P08473 1/20 0.37
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
OXTR P30559 2/20 0.36
AVPR1A P37288 2/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
ESR2 Q92731 1/20 0.36
PTPN1 P18031 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278807 0.99 ACHE (0.43) ACHEITGB1ITGA4MYCWDR5
SCHEMBL8813977 0.91 ABL1 (0.41) ACHEITGB1ITGA4MYCWDR5
SCHEMBL2311 0.84 ITGB1 (0.43) ACHEITGB1ITGA4MYCWDR5
SCHEMBL2563 0.83 ITGB1 (0.42) ACHEITGB1ITGA4MYCWDR5
SCHEMBL8808660 0.83 KCNH2 (0.36) ACHEALDH1A1GAAL3MBTL1CD274
SCHEMBL8808945 0.83 S1PR1 (0.34) ACHEITGB1ITGA4MYCWDR5
SCHEMBL8808908 0.83 MAOB (0.39) ACHEITGB1ITGA4MYCWDR5
SCHEMBL8806612 0.82 MAOB (0.38) ACHEITGB1ITGA4MYCWDR5
SCHEMBL7270209 0.77 LTB4R2 (0.45) ACHEITGB1ITGA4MYCWDR5
SCHEMBL8485794 0.76 ABL1 (0.42) ACHEITGB1ITGA4MYCWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed