SCHEMBL8808945

SCHEMBL8808945

CCOC(=O)OC1(CNCc2ccc3sc(-c4ccccc4C#N)cc3c2)CCCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.34
HDAC1 Q13547 3/20 0.34
ACHE P22303 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CD274 Q9NZQ7 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
METTL3 Q86U44 2/20 0.31
PRKCQ Q04759 1/20 0.31
PRKCD Q05655 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
METTL14 Q9HCE5 1/20 0.31
NLRP3 Q96P20 1/20 0.30
MYC P01106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9079126 0.87 S1PR1 (0.35) S1PR1HDAC1ACHEALDH1A1KDM4E
SCHEMBL8813977 0.85 ABL1 (0.41) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL7280200 0.83 ACHE (0.44) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL8808660 0.82 KCNH2 (0.36) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL8808908 0.82 MAOB (0.39) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL7278807 0.82 ACHE (0.43) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL8806612 0.82 MAOB (0.38) ACHEALDH1A1KDM4EHSD17B10CD274
SCHEMBL8806815 0.81 ACHE (0.34) ACHE
SCHEMBL8807911 0.74 TP53 (0.33) ACHEALDH1A1KDM4EHSD17B10GAA
SCHEMBL8911282 0.72 LTB4R2 (0.34) ACHEALDH1A1KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528762-B1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
EP-0528762-A1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA-GEIGY AG (CH) 1993-02-24 EP disclosed