SCHEMBL8808908

SCHEMBL8808908

CCOC(=O)OC1(CNCc2ccc3oc(-c4ccccc4C#N)cc3c2)CCCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.39
MAOA P21397 3/20 0.39
PRKCQ Q04759 4/20 0.35
PRKCD Q05655 4/20 0.35
CD274 Q9NZQ7 2/20 0.33
PDCD1 Q15116 1/20 0.33
MYC P01106 1/20 0.33
WDR5 P61964 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
ACHE P22303 1/20 0.32
JAK2 O60674 1/20 0.32
JAK3 P52333 1/20 0.32
CYP3A4 P08684 1/20 0.32
CA12 O43570 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8806612 0.99 MAOB (0.38) MAOBMAOAPRKCQPRKCDCD274
SCHEMBL8487461 0.87 MAOB (0.40) MAOBMAOAPRKCQPRKCDMYC
SCHEMBL8482882 0.86 MAOB (0.39) MAOBMAOAPRKCQPRKCDMYC
SCHEMBL8813977 0.85 ABL1 (0.41) CD274MYCWDR5KDM4EALDH1A1
SCHEMBL7280200 0.83 ACHE (0.44) CD274MYCWDR5KDM4EALDH1A1
SCHEMBL8808945 0.82 S1PR1 (0.34) PRKCQPRKCDCD274MYCWDR5
SCHEMBL8808660 0.82 KCNH2 (0.36) CD274KDM4EALDH1A1HSD17B10HRH3
SCHEMBL7278807 0.82 ACHE (0.43) CD274MYCWDR5KDM4EALDH1A1
SCHEMBL8811173 0.81 S1PR1 (0.34) MAOBMAOAPRKCQPRKCDMYC
SCHEMBL8808994 0.81 S1PR1 (0.34) MAOBMAOAPRKCQPRKCDMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528762-B1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA GEIGY AG (CH) 1997-05-07 EP disclosed
EP-0528762-A1 N-acyl-N-heterocyclyl- or naphthyl-alkyl amino acids as angiotensin II antagonists CIBA-GEIGY AG (CH) 1993-02-24 EP disclosed