SCHEMBL7280246

SCHEMBL7280246

CCCCCCCCOc1ccc(C(=O)ON2C(=O)c3ccccc3C2=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.55
TSHR P16473 1/20 0.55
PLA2G4B P0C869 5/20 0.53
RARB P10826 3/20 0.51
NPC1 O15118 2/20 0.50
LMNA P02545 2/20 0.50
NFKB1 P19838 1/20 0.50
NFKB2 Q00653 1/20 0.50
RELA Q04206 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PLA2G4A P47712 1/20 0.49
RECQL P46063 1/20 0.49
THRA P10827 1/20 0.48
THRB P10828 1/20 0.48
PTPN11 Q06124 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14774009 0.84 SMPD1 (0.50) RARBNPC1CYP1A2CYP2C9CYP2C19
SCHEMBL13604062 0.84 THRA (0.48) RARBTHRATHRB
SCHEMBL3683047 0.82 TP53 (0.57) TP53TSHRPLA2G4BRARBNPC1
SCHEMBL16142447 0.79 ALDH1A1 (0.50) NPC1SMN1; SMN2CYP1A2CYP2C9
SCHEMBL7271786 0.79 TP53 (0.53) TP53TSHRPLA2G4BRARBNPC1
SCHEMBL7280580 0.79 RARB (0.60) TP53TSHRPLA2G4BRARBNPC1
SCHEMBL3067042 0.79 RARB (0.60) TP53TSHRPLA2G4BRARBNPC1
SCHEMBL28548628 0.78 GAA (0.60) TP53NPC1SMN1; SMN2RECQLCYP1A2
SCHEMBL13479793 0.78 ALDH1A1 (0.55) SMN1; SMN2CYP1A2CYP2C9
SCHEMBL878923 0.78 HPGD (0.52) TP53TSHRPLA2G4BSMN1; SMN2THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-H1638-H CYCLIC HEXAPEPTIDE FURUTA TAKAHISA (JP) 1997-03-04 US disclosed
EP-0462531-B1 Cyclic polypeptide with antibiotic activity, process for its preparation and pure culture of a Coelomycetes strain FUJISAWA PHARMACEUTICAL CO (JP) 1996-10-02 EP disclosed
EP-0729974-A1 Cyclic polypeptide with antibiotic activity and a process for preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-09-04 EP disclosed
US-5376634-A Microbiocides FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-12-27 US disclosed
EP-0486011-A2 Pharmaceutical composition against Pneumocystis carinii FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-05-20 EP disclosed
EP-0462531-A2 Cyclic polypeptide with antibiotic activity, process for its preparation and pure culture of a Coelomycetes strain FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-27 EP disclosed