SCHEMBL7280302

SCHEMBL7280302

NCCc1ccc(OC[C@@H]2C[C@@H](CC(=O)O)C(=O)N2CCCc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
FFAR1 O14842 2/20 0.40
S1PR1 P21453 5/20 0.38
S1PR3 Q99500 2/20 0.38
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
SIGMAR1 Q99720 3/20 0.38
S1PR5 Q9H228 1/20 0.37
SSTR5 P35346 1/20 0.37
HTR2A P28223 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
HTR7 P34969 1/20 0.37
OPRM1 P35372 1/20 0.37
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL7277736 0.95 SIGMAR1 (0.41) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7284926 0.95 FFAR1 (0.41) ALDH1A1LMNAMAPTFFAR1S1PR1
Hydrochloric Acid SCHEMBL7274706 0.94 FFAR1 (0.40) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7284295 0.94 S1PR1 (0.40) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7275542 0.94 ALDH1A1 (0.40) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7274755 0.93 FFAR1 (0.41) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7280816 0.92 SSTR5 (0.43) FFAR1SSTR5LTA4H
SCHEMBL7272371 0.91 FFAR1 (0.41) ALDH1A1LMNAMAPTFFAR1S1PR1
Water SCHEMBL8882300 0.91 ITGB3 (0.38) ALDH1A1LMNAMAPTFFAR1S1PR1
SCHEMBL7274052 0.89 FFAR1 (0.43) FFAR1S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed