SCHEMBL7280596

SCHEMBL7280596

N[C@@H](Cc1ccc(F)nc1)C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.57
SLC7A5 Q01650 3/20 0.54
PTGS1 P23219 3/20 0.53
PKM P14618 2/20 0.53
ALPI P09923 1/20 0.53
XIAP P98170 1/20 0.53
HIF1A Q16665 3/20 0.50
ALOX15 P16050 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
GRB2 P62993 1/20 0.50
KDM4E B2RXH2 1/20 0.50
USP2 O75604 1/20 0.50
EGFR P00533 1/20 0.50
LCK P06239 1/20 0.50
FYN P06241 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
HTR2A P28223 1/20 0.50
PTGS2 P35354 1/20 0.50
RECQL P46063 1/20 0.50
PTPN1 P18031 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5291267 1.00 HSD17B10 (0.57) HSD17B10SLC7A5PTGS1PKMALPI
Trifluoroacetic Acid SCHEMBL27041676 0.93 GRB2 (0.58) HSD17B10SLC7A5PTGS1PKMALPI
SCHEMBL12629273 0.86 SLC1A1 (0.59) HSD17B10SLC7A5
SCHEMBL12762354 0.86 SLC1A1 (0.59) HSD17B10SLC7A5
SCHEMBL17054271 0.81 ALDH1A1 (0.45) HSD17B10PTGS2ALDH1A1
SCHEMBL4629770 0.81 CPB2 (0.63) HSD17B10SLC7A5PTGS1PKMALPI
SCHEMBL15314368 0.81 CPB2 (0.63) HSD17B10SLC7A5PTGS1PKMALPI
SCHEMBL229044 0.81 SLC7A5 (0.61) HSD17B10SLC7A5PTGS1PKMALPI
SCHEMBL26008176 0.81 CPB2 (0.63) HSD17B10SLC7A5PTGS1PKMALPI
SCHEMBL19704241 0.81 SLC7A5 (0.61) HSD17B10SLC7A5PTGS1PKMALPI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0073143-A2 Novel complex amido and imido derivatives of carboxyalkyl peptides and thioethers and ethers of peptides Ryan, James Walter (US) 1983-03-02 EP disclosed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed