SCHEMBL7280953

SCHEMBL7280953

N#Cc1ccc(-c2ccc(OC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)c(F)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.40
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
HTR2A P28223 1/20 0.37
HRH1 P35367 1/20 0.37
OPRM1 P35372 1/20 0.37
PPARD Q03181 3/20 0.36
FFAR1 O14842 2/20 0.36
ABCB1 P08183 1/20 0.36
HPGD P15428 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
PPARA Q07869 2/20 0.34
ALDH1A1 P00352 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FFAR4 Q5NUL3 2/20 0.34
NAMPT P43490 1/20 0.34
EP300 Q09472 2/20 0.34
SLK Q9H2G2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274966 0.92 HRH3 (0.40) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7274473 0.90 HTR1A (0.37) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7281974 0.90 MRGPRX4 (0.40) HRH3HTR1ADRD4HTR2AHRH1
Water SCHEMBL7281153 0.88 ITGB3 (0.41) OPRM1
SCHEMBL7275504 0.88 ABCB1 (0.45) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7276469 0.88 ABCB1 (0.45) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7282767 0.88 HRH3 (0.40) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7273894 0.88 HTR1A (0.35) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7273402 0.86 ABCB1 (0.44) HRH3HTR1ADRD4HTR2AHRH1
SCHEMBL7283417 0.85 HTR1A (0.37) HTR1ADRD4HTR2AHRH1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed