Bicarbonate

Bicarbonate

SCHEMBL7284102

Brc1ccc(C2CCC2)cc1.O=C(O)O.O=C(O)O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HDAC1 Q13547 1/20 0.52
HAO1 Q9UJM8 1/20 0.45
ACMSD Q8TDX5 2/20 0.44
ESR2 Q92731 6/20 0.44
HTT P42858 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GLA P06280 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL7273236 1.00 HDAC8 (0.52) HDAC8HDAC6HDAC1HAO1ACMSD
SCHEMBL11481277 0.92 HDAC8 (0.49) HDAC8HDAC6HDAC1HAO1ACMSD
SCHEMBL233178 0.89 ESR2 (0.47) HDAC8HDAC6HDAC1ESR2CYP3A4
Formic Acid SCHEMBL27517069 0.86 HDAC8 (0.46) HDAC8HDAC6HDAC1HAO1ESR2
SCHEMBL3575917 0.84 HDAC8 (0.50) HDAC8HDAC6HDAC1ESR2HTT
Cyanide SCHEMBL27788638 0.83 ESR2 (0.42) HDAC8HDAC6HDAC1ESR2CYP3A4
SCHEMBL17061138 0.82 HDAC8 (0.48) HDAC8HDAC6HDAC1HAO1ESR2
SCHEMBL126116 0.82 HDAC8 (0.48) HDAC8HDAC6HDAC1HAO1ESR2
SCHEMBL21609716 0.82 HDAC8 (0.48) HDAC8HDAC6HDAC1HAO1ESR2
SCHEMBL30056544 0.82 HDAC8 (0.48) HDAC8HDAC6HDAC1HAO1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed