SCHEMBL7284160

SCHEMBL7284160

CC(C)(C)OC(=O)NCCCC(=O)NC[C@@H]1CN(CCCc2ccccc2)C(=O)[C@H]1CC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.54
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
POLB P06746 1/20 0.42
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
HDAC4 P56524 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
CYP3A4 P08684 1/20 0.40
SIRT5 Q9NXA8 1/20 0.39
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273086 0.97 SIGMAR1 (0.51) SIGMAR1CA1CA2POLBHDAC3
SCHEMBL7283106 0.97 SIGMAR1 (0.51) SIGMAR1CA1CA2POLBHDAC3
SCHEMBL7282882 0.84 POLB (0.41) POLBHDAC3HDAC1HDAC8HDAC6
SCHEMBL7281050 0.81 NAMPT (0.41) POLBHDAC3HDAC1HDAC8HDAC6
SCHEMBL7283550 0.81 NAMPT (0.41) POLBHDAC3HDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL7283160 0.81 POLB (0.42) SIGMAR1POLBHDAC3HDAC1HDAC8
Hydrochloric Acid SCHEMBL8882333 0.81 POLB (0.42) SIGMAR1POLBHDAC3HDAC1HDAC8
Trifluoroacetic Acid SCHEMBL8881152 0.80 SIGMAR1 (0.40) SIGMAR1POLBHDAC3HDAC1HDAC8
SCHEMBL7283478 0.80 SIGMAR1 (0.54) SIGMAR1CA1CA2HDAC3HDAC1
SCHEMBL7274726 0.78 SIGMAR1 (0.51) SIGMAR1CA1CA2HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed