SCHEMBL7273086

SCHEMBL7273086

CC(C)(C)OC(=O)NCCCCCC(=O)NC[C@@H]1CN(CCCc2ccccc2)C(=O)[C@H]1CC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.51
CYP3A4 P08684 1/20 0.45
POLB P06746 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CACNA1G O43497 1/20 0.39
NAMPT P43490 2/20 0.39
TPSAB1 Q15661 1/20 0.39
TPSD1 Q9BZJ3 1/20 0.39
TPSG1 Q9NRR2 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283106 1.00 SIGMAR1 (0.51) SIGMAR1CYP3A4POLBNPSR1HDAC3
SCHEMBL7284160 0.97 SIGMAR1 (0.54) SIGMAR1CYP3A4POLBHDAC3HDAC1
SCHEMBL7281050 0.85 NAMPT (0.41) POLBHDAC3HDAC1HDAC8HDAC6
SCHEMBL7283550 0.85 NAMPT (0.41) POLBHDAC3HDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL8882333 0.83 POLB (0.42) SIGMAR1POLBHDAC3HDAC1HDAC8
Hydrochloric Acid SCHEMBL7283160 0.83 POLB (0.42) SIGMAR1POLBHDAC3HDAC1HDAC8
SCHEMBL7282882 0.81 POLB (0.41) POLBHDAC3HDAC1HDAC8HDAC6
SCHEMBL7274594 0.81 SIGMAR1 (0.51) SIGMAR1CYP3A4NPSR1HDAC3HDAC1
SCHEMBL7273844 0.81 SIGMAR1 (0.51) SIGMAR1CYP3A4NPSR1HDAC3HDAC1
SCHEMBL7275131 0.81 SIGMAR1 (0.51) SIGMAR1CYP3A4NPSR1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed