SCHEMBL7286097

SCHEMBL7286097

CC(C)(C)OC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ncc(C#N)s3)cc2)NC1=O

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
BRD4 O60885 1/20 0.34
IRAK4 Q9NWZ3 6/20 0.33
GPR119 Q8TDV5 3/20 0.33
DPP4 P27487 5/20 0.32
FAP Q12884 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285264 0.84 ITGB3 (0.53) ITGB3ITGA2BBRD4GPR119DPP4
Hydrochloric Acid SCHEMBL7284606 0.84 ITGB3 (0.53) ITGB3ITGA2BIRAK4
SCHEMBL7285015 0.84 ITGB3 (0.49) ITGB3ITGA2BBRD4IRAK4GPR119
SCHEMBL7283463 0.84 ITGB3 (0.49) ITGB3ITGA2BBRD4IRAK4GPR119
SCHEMBL8884076 0.84 ITGB3 (0.52) ITGB3ITGA2BBRD4GPR119DPP4
SCHEMBL7277677 0.82 ITGB3 (0.46) ITGB3ITGA2BBRD4IRAK4GPR119
SCHEMBL7275877 0.82 ITGB3 (0.46) ITGB3ITGA2BBRD4IRAK4GPR119
SCHEMBL7323680 0.78 ITGB3 (0.47) ITGB3ITGA2BGPR119
SCHEMBL7318086 0.78 ITGB3 (0.47) ITGB3ITGA2BIRAK4
SCHEMBL7277406 0.77 ITGB3 (0.47) ITGB3ITGA2BIRAK4GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed