SCHEMBL7285138

SCHEMBL7285138

COc1ccc(CCNC(=O)CCCCC(=O)O)c(F)c1OC

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 1/20 0.49
HPGD P15428 1/20 0.46
CNR1 P21554 2/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273517 0.90 HPGD (0.58) PTGER1HPGDMEN1KMT2ACYP1A2
SCHEMBL9786060 0.85 KDM4E (0.48) HPGDCNR1MEN1KMT2ACYP1A2
SCHEMBL7292858 0.83 HPGD (0.54) HPGD
SCHEMBL7366498 0.82 POLB (0.51) PTGER1MAPTPOLBKDM4E
SCHEMBL12192721 0.81 PTGER1 (0.50) PTGER1HPGDKDM4E
SCHEMBL9786061 0.80 SLC2A1 (0.52) HPGDCNR1MEN1KMT2ACYP1A2
SCHEMBL7293605 0.79 SLC2A1 (0.58) MEN1KMT2A
SCHEMBL7279723 0.79 HPGD (0.61) HPGDMEN1KMT2ACYP1A2CYP3A4
SCHEMBL7286269 0.77 ALDH1A1 (0.57) MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL7283066 0.77 MEN1 (0.59) HPGDMEN1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0223598-B1 CATECHOLAMINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS THEREOF FISONS plc (GB) 1991-06-12 EP disclosed
US-4939147-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC. (GB) 1990-07-03 US disclosed
US-4922022-A Substituted 3,4-dihydroxy phenylethylamino compounds FISONS PLC (GB) 1990-05-01 US disclosed
US-4883804-A Aromatic compounds FISONS PLC (GB) 1989-11-28 US disclosed
EP-0223598-A2 Catecholamine derivatives, processes for their preparation and pharmaceutical compositions thereof FISONS plc (GB) 1987-05-27 EP disclosed