SCHEMBL7285481

SCHEMBL7285481

COC(=O)c1ccc2n[c]oc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.47
ALOX15 P16050 2/20 0.47
CREBBP Q92793 1/20 0.46
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CA12 O43570 2/20 0.45
CA7 P43166 2/20 0.45
CA9 Q16790 2/20 0.45
CA14 Q9ULX7 2/20 0.45
XDH P47989 1/20 0.45
PSMB8 P28062 1/20 0.44
KDM4E B2RXH2 6/20 0.43
MAPT P10636 6/20 0.43
ALDH1A1 P00352 5/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
HPGD P15428 4/20 0.43
HSD17B10 Q99714 4/20 0.43
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
ATM Q13315 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5728015 0.88 KDM4E (0.45) HTTALOX15CREBBPCA1CA2
SCHEMBL27295800 0.73 TAS1R3 (0.56) HTTALOX15CREBBPCA1CA2
SCHEMBL1680291 0.72 ALDH1A1 (0.59) HTTALOX15CREBBPPSMB8KDM4E
SCHEMBL11781256 0.72 CA12 (0.49) CA1CA2CA12CA7CA9
SCHEMBL28562583 0.71 MAPT (0.54) HTTALOX15CREBBPCA1CA2
SCHEMBL7474034 0.71 HTT (0.46) HTTALOX15CA1CA2CA12
SCHEMBL2361382 0.71 MAPT (0.54) HTTALOX15CREBBPCA1CA2
SCHEMBL1101431 0.71 MAPT (0.54) HTTALOX15CREBBPCA1CA2
SCHEMBL31430581 0.71 MAPT (0.54) HTTALOX15CREBBPCA1CA2
SCHEMBL70757 0.69 CREBBP (0.57) HTTALOX15CREBBPCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0291234-B1 Peptidic human leukocyte elastase (HLE) inhibitors ZENECA INC (US) 1994-03-23 EP disclosed
US-5164371-A HETEROCYCLIC KETONES ICI AMERICAS INC. (US) 1992-11-17 US disclosed
CN-1037519-A HETEROCYCLIC KETONES ICI AMERICA INC (US) 1989-11-29 CN disclosed
EP-0291234-A2 Peptidic human leukocyte elastase (HLE) inhibitors ZENECA INC. (US) 1988-11-17 EP disclosed