SCHEMBL7286109

SCHEMBL7286109

COC(=O)c1ccc2cc(S(=O)(=O)C(F)(F)F)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPAS1 Q99814 1/20 0.48
PLAU P00749 4/20 0.48
POLB P06746 2/20 0.48
PTPN11 Q06124 1/20 0.48
NOTUM Q6P988 1/20 0.46
LCK P06239 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CYP2C9 P11712 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HGFAC Q04756 1/20 0.44
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PLAT P00750 1/20 0.43
CYP19A1 P11511 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29144762 0.84 CA1 (0.56) POLBCA12CA1CA2CA9
SCHEMBL28667831 0.82 POLB (0.51) EPAS1POLBKMT2ACA12CA1
SCHEMBL18513397 0.81 PTPN1 (0.53) EPAS1POLBMEN1KMT2ACA12
SCHEMBL22662913 0.80 PTPN11 (0.51) PLAUPOLBPTPN11LCKCA12
SCHEMBL3316267 0.79 STS (0.49) PLAUPTPN11NOTUMLCKCA12
SCHEMBL69025 0.79 PTPN11 (0.68) PLAUPTPN11LCKMEN1KMT2A
SCHEMBL29365729 0.79 PTPN11 (0.68) PLAUPTPN11LCKMEN1KMT2A
SCHEMBL732953 0.78 NOTUM (0.50) EPAS1POLBNOTUMMEN1KMT2A
SCHEMBL27367160 0.78 CYP2C9 (0.52) PLAUPOLBPTPN11LCKCYP2C9
SCHEMBL6002200 0.77 EPAS1 (0.49) EPAS1NOTUMMEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0744406-B1 Cyclic peptide antifungal agents LILLY CO ELI (US) 2002-09-04 EP disclosed
US-5629290-A Cyclic peptide antifungal agents ELI LILLY AND COMPANY (US) 1997-05-13 US disclosed
EP-0744406-A2 Cyclic peptide antifungal agents ELI LILLY AND COMPANY (US) 1996-11-27 EP disclosed