SCHEMBL7287239

SCHEMBL7287239

COC(=O)C[C@@H]1C[C@@H](CNC(=O)N2CCc3ccc(C#N)cc3C2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.49
DRD2 P14416 7/20 0.37
DRD3 P35462 5/20 0.37
DRD4 P21917 3/20 0.37
OPRM1 P35372 3/20 0.37
GPR183 P32249 1/20 0.36
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35
HRH1 P35367 1/20 0.35
MTNR1A P48039 1/20 0.34
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7284819 0.96 NAMPT (0.45) NAMPTDRD2DRD3DRD4OPRM1
SCHEMBL7275479 0.93 NAMPT (0.52) NAMPTDRD2DRD3DRD4OPRM1
SCHEMBL7286583 0.89 NAMPT (0.47) NAMPTDRD2DRD3DRD4OPRM1
Hydrochloric Acid SCHEMBL7335027 0.86 ITGB3 (0.37) NAMPTGPR183
Hydrochloric Acid SCHEMBL7277393 0.86 ITGB3 (0.37) NAMPTGPR183
SCHEMBL7284718 0.82 HTR1A (0.42) NAMPTDRD2DRD3DRD4HTR1A
SCHEMBL7273026 0.81 NAMPT (0.40) NAMPTDRD2DRD3DRD4OPRM1
Hydrochloric Acid SCHEMBL7276227 0.81 ITGB3 (0.36) OPRM1MTNR1A
SCHEMBL7274972 0.81 NAMPT (0.40) NAMPTDRD2DRD3DRD4HTR1A
SCHEMBL7283192 0.80 NR1H2 (0.40) NAMPTOPRM1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed