SCHEMBL7287458

SCHEMBL7287458

O=C1Nc2ccccc2SCC1c1ccc(Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
HSD17B10 Q99714 3/20 0.40
KDM4E B2RXH2 1/20 0.40
USP2 O75604 1/20 0.40
ESR1 P03372 1/20 0.40
POLB P06746 1/20 0.40
THRB P10828 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
PTPN7 P35236 1/20 0.40
RECQL P46063 1/20 0.40
ESR2 Q92731 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MAPK1 P28482 2/20 0.39
TNKS2 Q9H2K2 1/20 0.39
ACHE P22303 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7287889 0.82 MAPT (0.47) ALDH1A1MEN1KMT2ANPC1HSD17B10
SCHEMBL7285051 0.82 DDB1 (0.50) ALDH1A1MEN1KMT2ANPC1HSD17B10
SCHEMBL9765801 0.81 MAPT (0.43) ALDH1A1MEN1KMT2AHSD17B10ALOX15
SCHEMBL7289668 0.77 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AHSD17B10KDM4E
SCHEMBL10650323 0.75 HSD17B10 (0.49) ALDH1A1MEN1KMT2ANPC1HSD17B10
SCHEMBL7296419 0.74 DDB1 (0.55) ALDH1A1MEN1KMT2ANPC1KDM4E
SCHEMBL7298642 0.74 MEN1 (0.43) ALDH1A1MEN1KMT2AHSD17B10KDM4E
SCHEMBL8905187 0.72 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ANPC1HSD17B10
SCHEMBL8853352 0.72 ALDH1A1 (0.66) ALDH1A1MEN1KMT2ANPC1HSD17B10
SCHEMBL4495147 0.72 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ANPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0394101-B1 Benzothiazepine derivatives, process for their preparation and thereby obtained intermediates, their use as medicines and compositions containing them ROUSSEL UCLAF (FR) 1994-08-24 EP disclosed
US-5063225-A Antiarrhythmia ROUSSEL UCLAF (FR) 1991-11-05 US disclosed
EP-0394101-A1 Benzothiazepine derivatives, process for their preparation and thereby obtained intermediates, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1990-10-24 EP disclosed