SCHEMBL11484008

SCHEMBL11484008

COc1ccc2c(c1)OCC(CO)O2

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.56
MAPT P10636 3/20 0.49
GAA P10253 1/20 0.49
FFAR1 O14842 2/20 0.47
ALOX5 P09917 2/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
ADRA1D P25100 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29444764 0.94 MTNR1A (0.63) MTNR1AMAPTGAAFFAR1ALOX5
SCHEMBL1870686 0.94 MTNR1A (0.63) MTNR1AMAPTGAAFFAR1ALOX5
SCHEMBL6982719 0.94 MTNR1A (0.63) MTNR1AMAPTGAAFFAR1ALOX5
SCHEMBL28716707 0.83 FFAR1 (0.54) MTNR1AMAPTGAAFFAR1ALDH1A1
SCHEMBL28720097 0.83 FFAR1 (0.54) MTNR1AMAPTGAAFFAR1ALDH1A1
SCHEMBL11232203 0.82 MTNR1A (0.57) MTNR1AMAPTGAAFFAR1ALOX5
SCHEMBL9696456 0.81 ALOX5 (0.65) ALOX5ADRA1DADRA1AADRA1BADRB2
SCHEMBL8288367 0.80 CA2 (0.51) MTNR1AGAA
SCHEMBL1107090 0.80 CA2 (0.51) MTNR1AGAA
SCHEMBL1107087 0.80 CA2 (0.51) MTNR1AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4188390-A Antihypertensive 4-amino-2-[4-(1,4-benzodioxan-2-carbonyl) piperazin-1-yl or homopiperazin-1-yl]quinazolines PFIZER INC. (US) 1980-02-12 US disclosed