SCHEMBL7288172

SCHEMBL7288172

O=C(O)c1cnc2c(Br)csc2c1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 6/20 0.40
TSHR P16473 1/20 0.38
KDM4E B2RXH2 1/20 0.38
AKR1C4 P17516 2/20 0.37
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
AKR1C1 Q04828 2/20 0.37
PTPN1 P18031 2/20 0.34
CHEK1 O14757 1/20 0.34
LIMK1 P53667 1/20 0.34
DYRK1A Q13627 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
TTR P02766 1/20 0.32
HAVCR2 Q8TDQ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PTPN2 P17706 1/20 0.32
PTPN6 P29350 1/20 0.32
GABRP O00591 1/20 0.31
GABRD O14764 1/20 0.31
GABRA1 P14867 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279018 0.82 PDPK1 (0.41) GPR35KDM4EALDH1A1GABRPGABRD
SCHEMBL10578245 0.76 TSHR (0.40) TSHRGABRPGABRDGABRA1GABRB1
SCHEMBL16515634 0.75 KDM4E (0.45) GPR35TSHRKDM4EALDH1A1
SCHEMBL31400054 0.71 PDPK1 (0.39) KDM4EAKR1C3AKR1C2AKR1C1PTPN1
SCHEMBL31128943 0.69 TSHR (0.37) GPR35TSHRKDM4ECHEK1LIMK1
SCHEMBL4904323 0.69 AKR1C3 (0.36) GPR35TSHRKDM4EAKR1C4AKR1C3
SCHEMBL4543435 0.68 GPR35 (0.41) GPR35KDM4ECHEK1LIMK1DYRK1A
SCHEMBL15053880 0.67 EPRS1 (0.48) KDM4EAKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL15054611 0.67 KDM4E (0.41) TSHRKDM4EAKR1C4AKR1C3AKR1C2
SCHEMBL2207338 0.67 AKR1C3 (0.41) TSHRKDM4EAKR1C4AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560348-B1 Thieno 3,2-b pyridine derivatives for the treatment of gastrointestinal disorders MITSUBISHI CHEM CORP (JP) 2002-07-10 EP disclosed
US-5352685-A Gastrointestinal disorders MITSUBISHI KASEI CORPORATION (JP) 1994-10-04 US disclosed
EP-0560348-A1 Thieno 3,2-b pyridine derivatives for the treatment of gastrointestinal disorders Mitsubishi Chemical Corporation (JP) 1993-09-15 EP disclosed