SCHEMBL7289449

SCHEMBL7289449

COc1cc2c(cc1OC)C(C)(C1CCN(CCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC1)OCC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.45
SIGMAR1 Q99720 1/20 0.40
DRD2 P14416 2/20 0.38
DRD4 P21917 2/20 0.38
DRD3 P35462 2/20 0.38
CACNA1F O60840 1/20 0.38
HTR1A P08908 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
DRD5 P21918 1/20 0.38
HRH2 P25021 1/20 0.38
ADRA1D P25100 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
ADRA1B P35368 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL9147570 0.94 KCNH2 (0.42) KCNH2DRD2DRD4DRD3CACNA1F
Fumaric Acid SCHEMBL9147578 0.94 KCNH2 (0.42) KCNH2DRD2DRD4DRD3CACNA1F
SCHEMBL7292071 0.92 SIGMAR1 (0.49) SIGMAR1
SCHEMBL7299887 0.88 SLC6A4 (0.42) KCNH2SIGMAR1OPRM1OPRK1SLC6A3
SCHEMBL7289129 0.86 SLC6A4 (0.46) SIGMAR1SLC6A3
SCHEMBL7291347 0.85 DRD2 (0.42) DRD2DRD4DRD3SLC6A3
SCHEMBL7291776 0.81 KCNH2 (0.47) KCNH2DRD2DRD4DRD3CACNA1F
SCHEMBL7298566 0.79 SLC6A2 (0.43) SIGMAR1SLC6A3
SCHEMBL7322676 0.75 KCNH2 (0.42) KCNH2DRD2DRD4DRD3
SCHEMBL7292905 0.74 KCNH2 (0.54) KCNH2DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458387-B1 Isochromane derivatives AKZO NOBEL NV (NL) 1996-07-03 EP disclosed
US-5393759-A Isochromane derivatives AKZO N.V. (NL) 1995-02-28 US disclosed
US-5238939-A Isochromane derivatives AKZO N.V. (NL) 1993-08-24 US disclosed
EP-0458387-A1 Isochromane derivatives Akzo Nobel N.V. (NL) 1991-11-27 EP disclosed