SCHEMBL7322676

SCHEMBL7322676

CCC1(CCN2CCN(CCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2)OCCc2cc(OC)c(OC)cc21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.42
CCR2 P41597 2/20 0.38
KMT2A Q03164 1/20 0.36
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
ABCB1 P08183 1/20 0.35
TACR1 P25103 1/20 0.35
FAAH O00519 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
MTOR P42345 1/20 0.35
RAB9A P51151 1/20 0.35
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7291776 0.95 KCNH2 (0.47) KCNH2KMT2ADRD2DRD4DRD3
Fumaric Acid SCHEMBL9149650 0.93 CCR2 (0.39) KCNH2CCR2FAAHCYP3A4CYP2D6
Fumaric Acid SCHEMBL9149646 0.93 CCR2 (0.39) KCNH2CCR2FAAHCYP3A4CYP2D6
SCHEMBL7292958 0.93 KCNH2 (0.38) KCNH2CCR2KMT2ADRD2DRD4
SCHEMBL7294243 0.88 SIGMAR1 (0.43)
SCHEMBL7289973 0.87 SLC6A3 (0.44) DRD2DRD4DRD3
SCHEMBL7289109 0.86 SIGMAR1 (0.39) KCNH2DRD2DRD4DRD3
SCHEMBL7291484 0.83 MAOA (0.37) DRD4ABCB1CYP2D6TSHR
SCHEMBL7298864 0.83 CCR2 (0.44) KCNH2CCR2KMT2ADRD2DRD3
SCHEMBL9490288 0.83 CCR2 (0.34) KCNH2CCR2TACR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458387-B1 Isochromane derivatives AKZO NOBEL NV (NL) 1996-07-03 EP disclosed
US-5393759-A Isochromane derivatives AKZO N.V. (NL) 1995-02-28 US disclosed
US-5238939-A Isochromane derivatives AKZO N.V. (NL) 1993-08-24 US disclosed
EP-0458387-A1 Isochromane derivatives Akzo Nobel N.V. (NL) 1991-11-27 EP disclosed