SCHEMBL7289822

SCHEMBL7289822

C=C[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)C

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
KLK5 Q9Y337 1/20 0.51
CTSS P25774 3/20 0.50
CTSK P43235 2/20 0.50
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
APP P05067 1/20 0.49
BACE1 P56817 2/20 0.48
PSEN1 P49768 3/20 0.47
PSEN2 P49810 3/20 0.47
APH1B Q8WW43 3/20 0.47
NCSTN Q92542 3/20 0.47
APH1A Q96BI3 3/20 0.47
PSENEN Q9NZ42 3/20 0.47
REN P00797 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9078755 0.90 CTSB (0.57) ATMMEN1KMT2AKLK5CTSS
SCHEMBL9017588 0.90 CTSB (0.57) ATMMEN1KMT2AKLK5CTSS
SCHEMBL20204825 0.90 CTSB (0.57) ATMMEN1KMT2AKLK5CTSS
SCHEMBL1207885 0.88 ATM (0.57) ATMKLK5CTSSCTSKCTSL
SCHEMBL5732519 0.88 ATM (0.57) ATMKLK5CTSSCTSKCTSL
SCHEMBL13937947 0.88 ATM (0.57) ATMKLK5CTSSCTSKCTSL
SCHEMBL29602242 0.82 KMT2A (0.67) ATMMEN1KMT2AKLK5CTSS
SCHEMBL8130179 0.82 KMT2A (0.67) ATMMEN1KMT2AKLK5CTSS
SCHEMBL8539393 0.82 KLK5 (0.52) ATMMEN1KMT2AKLK5CTSS
SCHEMBL8542012 0.81 CYP3A4 (0.59) ATMMEN1KMT2AKLK5CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605926-A PROPHYLAXIS BAYER AKTIENGESELLSCHAFT (DE) 1997-02-25 US disclosed
US-5430151-A Treatment of aids, pneumonia, caprine arthritis encephalitis, leukemia and immmunodeficiency BAYER AKTIENGESELLSCHAFT (DE) 1995-07-04 US disclosed
US-5204471-A α-trifluoromethyl-substituted, saturated bicyclic amines BAYER AKTIENGESELLSCHAFT (DE) 1993-04-20 US disclosed
EP-0528242-A2 Trifluoromethyl containing pseudopeptides BAYER AG (DE) 1993-02-24 EP disclosed
EP-0472077-A2 Phosphonate containing hydroxyethylamin- and norstatin-type pseudopeptides BAYER AG (DE) 1992-02-26 EP disclosed