SCHEMBL8542012

SCHEMBL8542012

CC(C)[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CO)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.59
MAPK1 P28482 1/20 0.59
ATM Q13315 2/20 0.57
APP P05067 2/20 0.56
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
KLK5 Q9Y337 1/20 0.53
CTSS P25774 3/20 0.52
CTSK P43235 2/20 0.52
CTSL P07711 1/20 0.52
CTSB P07858 1/20 0.52
BACE1 P56817 2/20 0.49
PSEN1 P49768 2/20 0.49
PSEN2 P49810 2/20 0.49
APH1B Q8WW43 2/20 0.49
NCSTN Q92542 2/20 0.49
APH1A Q96BI3 2/20 0.49
PSENEN Q9NZ42 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532232 0.89 ATM (0.69) ATMAPPMEN1KMT2AKLK5
SCHEMBL271855 0.87 ATM (0.71) CYP3A4MAPK1ATMAPPKLK5
SCHEMBL1529562 0.87 ATM (0.71) CYP3A4MAPK1ATMAPPKLK5
SCHEMBL257912 0.87 ATM (0.71) CYP3A4MAPK1ATMAPPKLK5
SCHEMBL7349961 0.87 ATM (0.58) CYP3A4MAPK1ATMAPPKLK5
SCHEMBL13669577 0.85 CTSS (0.67) CYP3A4MAPK1ATMAPPCTSS
SCHEMBL7323342 0.84 CYP3A4 (0.60) CYP3A4MAPK1CTSSCTSKCTSL
SCHEMBL8130179 0.84 KMT2A (0.67) ATMAPPMEN1KMT2AKLK5
SCHEMBL29602242 0.84 KMT2A (0.67) ATMAPPMEN1KMT2AKLK5
SCHEMBL27413971 0.84 REN (0.63) CYP3A4MAPK1ATMCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0503561-B1 Method for the diastereoselective reductive pinacol coupling of homochiral alpha aminoaldehydes HOECHST AG (DE) 1998-10-28 EP disclosed
EP-0541946-B1 Process for diastereo selective reductive pinacol-coupling of homochiral alpha-aminoaldehydes HOECHST AG (DE) 1996-07-17 EP disclosed
US-5519113-A Process for the diastereoselective reductive pinacol coupling of homochiral α-aminoaldehydes HOECHST AKTIENGESELLSCHAFT (DE) 1996-05-21 US disclosed
US-5463124-A Treating with niobium trichloride-dimethoxyethane complex and simultaneously controlling all four corners of chirality HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-31 US disclosed
EP-0541946-A1 Process for diastereo selective reductive pinacol-coupling of homochiral alpha-aminoaldehydes HOECHST AKTIENGESELLSCHAFT (DE) 1993-05-19 EP disclosed
EP-0503561-A2 Method for the diastereoselective reductive pinacol coupling of homochiral alpha aminoaldehydes HOECHST AKTIENGESELLSCHAFT (DE) 1992-09-16 EP disclosed