SCHEMBL7289846

SCHEMBL7289846

CSc1ccc(NC(=O)CCl)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.73
NPC1 O15118 4/20 0.73
MITF O75030 2/20 0.73
XBP1 P17861 1/20 0.73
NPSR1 Q6W5P4 1/20 0.73
NOD2 Q9HC29 1/20 0.73
MAPT P10636 9/20 0.60
ALDH1A1 P00352 8/20 0.60
SMN1; SMN2 Q16637 6/20 0.60
KMT2A Q03164 5/20 0.60
HPGD P15428 2/20 0.60
OPRM1 P35372 1/20 0.60
OPRD1 P41143 1/20 0.60
JAK2 O60674 1/20 0.60
PKM P14618 1/20 0.56
HTT P42858 3/20 0.56
PRMT1 Q99873 1/20 0.56
LMNA P02545 6/20 0.51
KDM4E B2RXH2 2/20 0.51
MEN1 O00255 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10920656 0.85 NPC1 (1.00) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL9081388 0.84 NPC1 (0.76) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL13370416 0.83 KMT2A (0.65) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL13602760 0.83 ALDH1A1 (0.53) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL6390723 0.81 CA1 (0.54) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL7724959 0.81 ALDH1A1 (0.51) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL14799129 0.81 ALDH1A1 (0.56) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL11692587 0.80 MAPT (0.60) RAB9ANPC1MITFXBP1NPSR1
SCHEMBL4007599 0.80 MEN1 (0.74) RAB9ANPC1MAPTALDH1A1SMN1; SMN2
SCHEMBL7827838 0.79 CYP1A1 (0.64) RAB9ANPC1MAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed