SCHEMBL7292149

SCHEMBL7292149

CC1(C)C=C(n2cc(Cl)cc(Cl)c2=O)c2ncccc2O1

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.31
NPC1 O15118 1/20 0.30
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300229 0.89 NR4A2 (0.31)
SCHEMBL7300599 0.89
SCHEMBL7315149 0.86 L3MBTL1 (0.35) NPC1
SCHEMBL7288952 0.85 TDP1 (0.33) NPC1
SCHEMBL7375797 0.84 NPC1 (0.32) TNKSNPC1
SCHEMBL7313380 0.84 NPC1 (0.32) NPC1
SCHEMBL7372821 0.84 S100A4 (0.36) NPC1
SCHEMBL7374676 0.84 ALDH1A1 (0.38) NPC1
SCHEMBL7298334 0.82 TNKS (0.33) TNKS
SCHEMBL7299568 0.80 POLB (0.34) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308792-B1 AZACHROMANE DERIVATIVES MERCK PATENT GmbH (DE) 1993-07-28 EP disclosed
US-4931454-A Azachroman derivatives with effects on the cardiovascular system MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-06-05 US disclosed
EP-0308792-A2 Azachromane derivatives MERCK PATENT GmbH (DE) 1989-03-29 EP disclosed