SCHEMBL7292741

SCHEMBL7292741

CC(COC([NH])=O)Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
ATM Q13315 1/20 0.47
EGFR P00533 1/20 0.46
ALDH1A1 P00352 1/20 0.46
THRB P10828 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MAPT P10636 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CYP1A2 P05177 1/20 0.44
LMNA P02545 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAPK1 P28482 1/20 0.43
TSHR P16473 1/20 0.42
SRR Q9GZT4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5622799 0.86 NPC1 (0.53) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL16137501 0.84 ALDH1A1 (0.56) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL24073103 0.84 NPC1 (0.51) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL15247513 0.84 ALDH1A1 (0.56) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL10886546 0.84 ALDH1A1 (0.56) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL7260000 0.83 CYP3A4 (0.50) NPC1RAB9AATMEGFRALDH1A1
SCHEMBL22911682 0.83 PKM (0.54) NPC1RAB9AALDH1A1THRBCYP2C9
SCHEMBL7292748 0.83 PKM (0.54) NPC1RAB9AALDH1A1THRBCYP2C9
SCHEMBL17629341 0.81 ALDH1A1 (0.59) NPC1RAB9AEGFRALDH1A1MAPT
SCHEMBL8926076 0.81 NPC1 (0.49) NPC1RAB9AATMEGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
US-RE34722-E Antiulcer agents OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-09-06 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed
EP-0382185-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed
US-4578381-A ANTIULCER AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-03-25 US disclosed