SCHEMBL7293402

SCHEMBL7293402

COCCOCO[C@H]([C@H](CC1CCCCC1)NC(=O)OC(C)(C)C)[C@@H](O)CN(C)OC

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
REN P00797 14/20 0.38
CACNA1B Q00975 1/20 0.37
CTSD P07339 1/20 0.35
CTSE P14091 1/20 0.35
GAA P10253 1/20 0.33
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7293407 0.86 CTSS (0.39) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7280909 0.85 CTSS (0.40) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7281024 0.85 CTSS (0.40) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7281111 0.85 CTSK (0.48) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7291461 0.84 CTSS (0.43) CTSSCTSKRENCACNA1BCTSD
SCHEMBL10592277 0.84 CTSS (0.41) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7299478 0.84 CTSS (0.41) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7298823 0.81 CTSS (0.36) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7293395 0.80 CTSS (0.39) CTSSCTSKRENCACNA1BCTSD
SCHEMBL7293382 0.79 REN (0.37) CTSSCTSKRENCTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5268374-A Containing both amide and hydroxy groups ABBOTT LABORATORIES (US) 1993-12-07 US disclosed
EP-0437508-A1 NON-PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-07-24 EP disclosed
WO-1990003971-A1 NON-PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-04-19 WO disclosed
WO-1989010751-A1 FUNCTIONALIZED PEPTIDYL AMINODIOLS AND -TRIOLS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
EP-0341602-A2 Renin-inhibiting functionalized peptidyl aminodiols and - triols ABBOTT LABORATORIES (US) 1989-11-15 EP disclosed