SCHEMBL7295604

SCHEMBL7295604

O=c1[nH]c2nc[nH]c2c(=O)n1CC1CCCCC1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.59
PDE4A P27815 3/20 0.59
PDE4B Q07343 3/20 0.59
PDE4C Q08493 3/20 0.59
PDE4D Q08499 3/20 0.59
ADORA2B P29275 7/20 0.59
ADORA3 P0DMS8 6/20 0.59
MTOR P42345 8/20 0.48
PIK3CA P42336 1/20 0.48
GSK3A P49840 1/20 0.48
JAK2 O60674 1/20 0.48
JAK1 P23458 1/20 0.48
JAK3 P52333 1/20 0.48
ADORA1 P30542 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7295708 0.99 ADORA2A (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7296248 0.96 ADORA2A (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL6141778 0.93 ADORA2A (0.64) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL31366236 0.84 ADORA2A (0.59) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL29429682 0.80 ADORA2A (0.49) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27621962 0.80 ADORA2B (0.66) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL10978398 0.78 PDE4A (0.59) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7025705 0.77 ADORA2B (0.55) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27543834 0.76 ADORA2B (0.97) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7617653 0.76 ADORA2B (0.50) ADORA2AADORA2BADORA3MTORPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0389282-B1 Xanthinederivatives, process for their preparation and their pharmaceutical use SMITHKLINE BEECHAM PHARMA GMBH (DE) 2002-02-20 EP disclosed