SCHEMBL29429682

SCHEMBL29429682

O=c1[nH]c2nc[nH]c2c(=O)n1CC1CCC(O)(C(F)(F)F)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.49
PDE4A P27815 3/20 0.49
PDE4B Q07343 3/20 0.49
PDE4C Q08493 3/20 0.49
PDE4D Q08499 3/20 0.49
ADORA2B P29275 10/20 0.47
ADORA3 P0DMS8 8/20 0.47
ADORA1 P30542 3/20 0.45
GRIN1 Q05586 3/20 0.36
GRIN2B Q13224 3/20 0.36
MTOR P42345 2/20 0.34
PIK3CA P42336 1/20 0.34
GSK3A P49840 1/20 0.34
CD38 P28907 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141778 0.83 ADORA2A (0.64) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7296248 0.81 ADORA2A (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7295708 0.81 ADORA2A (0.61) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL7295604 0.80 ADORA2A (0.59) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL31366236 0.75 ADORA2A (0.59) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL27621962 0.74 ADORA2B (0.66) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL30025357 0.72 ADORA2A (0.66) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL5515444 0.70 ADORA2A (0.71) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL31065356 0.69 ADORA2A (0.58) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL4602969 0.68 ADORA2B (0.73) ADORA2APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49128-E1 Hydroxyl purine compounds and applications thereof Guangdong Raynovent Biotech Co., Ltd. (CN) 2022-07-12 US disclosed
EP-3205652-B1 HYDROXYL PURINE COMPOUNDS AND APPLICATIONS THEREOF GUANGDONG RAYNOVENT BIOTECH CO LTD (CN) 2022-03-09 EP disclosed