SCHEMBL7296197

SCHEMBL7296197

CC(C)(C)OC(=O)CCC(=O)O.c1ccc2c(c1)C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CD69 Q07108 2/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
NR4A2 P43354 1/20 0.39
NOTUM Q6P988 1/20 0.39
ELANE P08246 2/20 0.37
RBP4 P02753 1/20 0.37
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
MAPK1 P28482 1/20 0.37
EPHX2 P34913 1/20 0.37
NAMPT P43490 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL631111 0.82 EGLN1 (0.48) MAPK1KDM4E
SCHEMBL9755818 0.81 NOTUM (0.51) CD69CYP2C19NOTUMKDM4EMEN1
Cyclohexane SCHEMBL27625968 0.80 LMNA (0.44) EPHX2
Chloromethane SCHEMBL3415691 0.80 EGLN1 (0.46) MAPK1EPHX2KDM4E
Butane SCHEMBL2855608 0.76 FFAR3 (0.44) MEN1KMT2ATDP1
SCHEMBL2516124 0.76 NR4A2 (0.55) CYP2C19HIF1ANR4A2MAPK1KDM4E
SCHEMBL28117718 0.74 EGLN1 (0.42) MAPT
SCHEMBL9841927 0.74 CYP2D6 (0.38) CYP2C19MEN1KMT2A
SCHEMBL1380801 0.74 TDP1 (0.61) KDM4EMEN1MAPTKMT2ATDP1
SCHEMBL28412762 0.73 CYP2C19 (0.41) CYP2C19HIF1ANR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5164388-A Hypotensive agents, treatment of congestive heart failure ABBOTT LABORATORIES (US) 1992-11-17 US disclosed
EP-0439556-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1991-08-07 EP disclosed
WO-1990004917-A1 HETEROCYCLIC PEPTIDE RENIN INHIBITORS ABBOTT LABORATORIES (US) 1990-05-17 WO disclosed
EP-0365992-A1 Heterocyclic peptide renin inhibitors ABBOTT LABORATORIES (US) 1990-05-02 EP disclosed