SCHEMBL7297301

SCHEMBL7297301

Cc1cc2c(s1)SCCc1cc(=O)[nH]nc1-2

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
PDE3A Q14432 2/20 0.36
PDE4B Q07343 1/20 0.36
HRH3 Q9Y5N1 1/20 0.33
PDE3B Q13370 1/20 0.33
CA2 P00918 1/20 0.32
PLA2G10 O15496 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298398 0.83 GAA (0.39) GAAPDE3APDE4BHRH3PDE3B
SCHEMBL7287593 0.71 PDE3A (0.42) GAAPDE3APDE4BHRH3PDE3B
SCHEMBL7296693 0.69 ALDH1A1 (0.39) GAA
SCHEMBL10389368 0.68 GAA (0.46) GAAPDE3APDE4BHRH3PDE3B
SCHEMBL10388766 0.68 GAA (0.50) GAAPDE3APDE4BHRH3PDE3B
SCHEMBL7298799 0.66 CA2 (0.45) CA2
SCHEMBL4983802 0.65 GSR (0.51) GAAPDE3APDE4BHRH3PDE3B
SCHEMBL10341494 0.62 MEN1 (0.60) HRH3
SCHEMBL9039217 0.62 HPGD (0.45) GAACA2
SCHEMBL9039222 0.62 HPGD (0.45) GAACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0426018-B1 Thiophene compounds and their pharmaceutical uses YOSHITIOMI PHARMACEUTICAL IND (JP) 1997-08-27 EP disclosed
EP-0729960-A1 Thiophene compounds and their use as intermediates in the preparation of antianxiety drugs, hypnotics, antiepileptic drugs and nuotropics YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-09-04 EP disclosed
US-5329016-A Antianxiety, hypnotic agents, antiepileptic agents or nootropics YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-07-12 US disclosed
US-5175162-A Anxiolytic, antiepilepic agents YOSHITIOMI PHARMACEUTICAL INDUSTRIES LTD. (JP) 1992-12-29 US disclosed
EP-0426018-A2 Thiophene compounds and their pharmaceutical uses YOSHITIOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-05-08 EP disclosed