SCHEMBL7298263

SCHEMBL7298263

COC(=CC(=O)c1c(C)[nH]c(C)c1C(=O)O)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
MAPT P10636 6/20 0.43
NPSR1 Q6W5P4 2/20 0.43
TSHR P16473 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
HIF1A Q16665 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 5/20 0.42
RAB9A P51151 6/20 0.39
NPC1 O15118 4/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPK1 P28482 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298258 1.00 ALDH1A1 (0.43) ALDH1A1MAPTNPSR1TSHRCYP1A2
SCHEMBL12591107 0.74 CES2 (0.45) ALDH1A1MAPTTSHRLMNARAB9A
SCHEMBL7298648 0.72 ALDH1A1 (0.44) ALDH1A1MAPTTSHRLMNARAB9A
SCHEMBL7298652 0.72 ALDH1A1 (0.44) ALDH1A1MAPTTSHRLMNARAB9A
SCHEMBL19980208 0.68 ALDH1A1 (0.40) ALDH1A1MAPTTSHRHIF1ATDP1
SCHEMBL19980206 0.67 TSHR (0.41) ALDH1A1MAPTTSHRLMNARAB9A
SCHEMBL7291203 0.66 MAPT (0.61) ALDH1A1MAPTNPSR1TSHRCYP1A2
SCHEMBL23188930 0.66 TSHR (0.46) ALDH1A1MAPTTSHRCYP1A2LMNA
SCHEMBL21157019 0.66 ALDH1A1 (0.38) ALDH1A1MAPTTSHRHIF1ATDP1
SCHEMBL12591127 0.65 RAB9A (0.39) ALDH1A1MAPTTSHRLMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0300688-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them FISONS plc (GB) 1989-01-25 EP claimed
EP-0300688-A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them FISONS plc (GB) 1989-01-25 EP disclosed