SCHEMBL7298331

SCHEMBL7298331

CCCCOC(=O)CN1CCN(C(=O)[C@H](Cc2ccc(OC)cc2)NC(=O)OCc2ccccc2)[C@@H](CC(=O)OC)C1=O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.46
ITGA2B P08514 11/20 0.46
CTSL P07711 1/20 0.45
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
P2RX7 Q99572 4/20 0.44
ACE P12821 2/20 0.43
ACE2 Q9BYF1 2/20 0.43
HDAC8 Q9BY41 1/20 0.42
ITGAV P06756 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308737 0.92 P2RX7 (0.47) ITGB3ITGA2BCTSLCTSSCTSK
SCHEMBL7371887 0.90 P2RX7 (0.48) CTSLCTSKP2RX7HDAC8
SCHEMBL7371888 0.90 P2RX7 (0.48) CTSLCTSKP2RX7HDAC8
SCHEMBL7371886 0.90 P2RX7 (0.48) CTSLCTSKP2RX7HDAC8
SCHEMBL7303718 0.88 P2RX7 (0.43) ITGB3ITGA2BCTSLCTSSCTSK
SCHEMBL7301305 0.87 P2RX7 (0.43) ITGB3ITGA2BCTSLCTSSCTSK
SCHEMBL7297146 0.85 P2RX7 (0.49) ITGB3ITGA2BCTSLCTSKP2RX7
SCHEMBL7307823 0.84 P2RX7 (0.46) CTSLCTSSCTSKP2RX7
SCHEMBL7308051 0.83 ITGB3 (0.48) ITGB3ITGA2BCTSLCTSSCTSK
SCHEMBL7295570 0.82 ITGB3 (0.47) ITGB3ITGA2BCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643072-B1 2-Piperazinone compounds and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-02-24 EP disclosed
EP-0643072-A1 2-Piperazinone compounds and their use Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed