SCHEMBL7298570

SCHEMBL7298570

Cc1cncc(COC(=O)N[C@H](C(=O)O)C(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TYR P14679 3/20 0.48
GPR132 Q9UNW8 2/20 0.43
ECE1 P42892 2/20 0.42
MME P08473 1/20 0.42
CTSL P07711 4/20 0.41
CTSB P07858 3/20 0.41
CTSS P25774 3/20 0.41
CTSK P43235 2/20 0.41
ATM Q13315 1/20 0.39
CA1 P00915 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
CASP1 P29466 1/20 0.38
CASP3 P42574 1/20 0.38
CASP7 P55210 1/20 0.38
CASP9 P55211 1/20 0.38
CASP6 P55212 1/20 0.38
CASP8 Q14790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7298563 1.00 TYR (0.48) TYRGPR132ECE1MMECTSL
SCHEMBL7310825 0.85 TYR (0.46) TYRGPR132ECE1MMECTSL
SCHEMBL7310831 0.85 TYR (0.46) TYRGPR132ECE1MMECTSL
SCHEMBL23966258 0.81 POLB (0.53) TYRECE1MMECTSLCTSB
SCHEMBL8604954 0.80 CTSL (0.51) TYRECE1MMECTSLCTSB
SCHEMBL7269614 0.80 GPR132 (0.61) GPR132ECE1MMECTSLCTSB
SCHEMBL7269609 0.80 GPR132 (0.61) GPR132ECE1MMECTSLCTSB
SCHEMBL19607509 0.79 CTSL (0.55) TYRECE1MMECTSLCTSB
SCHEMBL7279121 0.79 CTSL (0.50) TYRECE1MMECTSLCTSB
SCHEMBL7279131 0.79 CTSL (0.50) TYRECE1MMECTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-B1 Retroviral protease inhibiting compounds ABBOTT LAB (US) 2000-10-04 EP disclosed
EP-0997459-A1 Intermediates for preparing retroviral protease inhibiting compounds Abbott Laboratories (US) 2000-05-03 EP disclosed
US-5837873-A PROTECTED OXYDIAMINES ABBOTT LABORATORIES (US) 1998-11-17 US disclosed
US-5648497-A Retroviral protease inhibiting compounds ABBOTT LABORAOTRIES (US) 1997-07-15 US disclosed
US-5616714-A PYRIDYL, THIAZOLYL-SUBSTITUTED AMINO ACID DERIVATIVES ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
US-5597926-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-01-28 US disclosed
US-5554783-A (2R, 3R, 4S, 5S)-3-ACETOXY-2,5-BIS/BENZYLOXYCARBONYLAMINO/ -4-BROMO-1,5-DIPHENYLHEXANE ABBOTT LABORATORIES (US) 1996-09-10 US disclosed
US-5541334-A TREATING HIV ABBOTT LABORATORIES (US) 1996-07-30 US disclosed
US-5354866-A Treating HIV infections ABBOTT LABORATORIES (US) 1994-10-11 US disclosed
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed