SCHEMBL7300495

SCHEMBL7300495

CC(C)CC(Cc1ccccc1)(Cc1ccccc1)O[PH](=O)OC(Cc1ccccc1)(Cc1ccccc1)CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.41
SLC6A2 P23975 3/20 0.36
TAAR1 Q96RJ0 3/20 0.36
LMNA P02545 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
HIF1A Q16665 1/20 0.33
CASR P41180 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
CTSK P43235 1/20 0.33
GAA P10253 1/20 0.33
FDPS P14324 1/20 0.33
MAOA P21397 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CYP2A6 P11509 1/20 0.32
ADORA2A P29274 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300498 0.87 TRPA1 (0.42) TRPA1SLC6A2TAAR1TSHRSMN1; SMN2
SCHEMBL7271496 0.84 SMN1; SMN2 (0.41) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL7273150 0.82 CTSK (0.41) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL11571239 0.72 TAAR1 (0.50) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL9312880 0.71 CYP1A2 (0.41) CASRCYP2A6HTR2A
SCHEMBL7273144 0.70 CTSK (0.43) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL27350008 0.70 TRPA1 (0.47) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL3363867 0.69 FDPS (0.46) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL7271492 0.69 SMN1; SMN2 (0.42) TRPA1SLC6A2TAAR1LMNACYP2D6
SCHEMBL1727267 0.69 TAAR1 (0.47) TRPA1SLC6A2TAAR1LMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35886-E ENDOTHELIN-CONVERTING ENZYME INHIBITOR TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-09-01 US disclosed
EP-0518299-B1 Phosphonic acid derivatives, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-08 EP disclosed
US-5330978-A Cardiovascular disorders, hypotensive agents, vasodilation TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-07-19 US disclosed
EP-0518299-A2 Phosphonic acid derivatives, production and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed