SCHEMBL7300635

SCHEMBL7300635

CC1(C)C=C(n2cc(N)ccc2=O)c2cccnc2O1

nearest known ligand 0.30

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300381 0.86 LMNA (0.31) TNKS
SCHEMBL7292763 0.83 SMN1; SMN2 (0.36) TNKS
SCHEMBL7297727 0.83 TDP1 (0.37)
SCHEMBL7299711 0.82 WEE1 (0.31)
SCHEMBL7379309 0.82 POLB (0.33)
SCHEMBL7299641 0.81 HRH4 (0.33)
SCHEMBL7300227 0.81 MEN1 (0.37)
SCHEMBL7298804 0.81 NPC1 (0.32) TNKS
SCHEMBL7378273 0.81 CDK8 (0.32)
SCHEMBL7348702 0.79 MEN1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308792-B1 AZACHROMANE DERIVATIVES MERCK PATENT GmbH (DE) 1993-07-28 EP disclosed
US-4931454-A Azachroman derivatives with effects on the cardiovascular system MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1990-06-05 US disclosed
EP-0308792-A2 Azachromane derivatives MERCK PATENT GmbH (DE) 1989-03-29 EP disclosed