SCHEMBL7300826

SCHEMBL7300826

CCCCC(NCC(CC(C)C)NC(=O)c1ccc(OC)cc1)C(=O)CSCc1ccco1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
HPGD P15428 5/20 0.41
POLB P06746 4/20 0.41
MAPT P10636 7/20 0.41
ALDH1A1 P00352 5/20 0.41
USP2 O75604 3/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
RECQL P46063 2/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442933 0.94 ALDH1A1 (0.44) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7306407 0.93 POLB (0.51) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7299096 0.91 ALDH1A1 (0.43) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7303801 0.91 ALDH1A1 (0.40) HPGDPOLBMAPTALDH1A1USP2
SCHEMBL7313603 0.90 ALDH1A1 (0.40) HPGDPOLBMAPTALDH1A1USP2
SCHEMBL7306946 0.89 ALDH1A1 (0.41) HPGDPOLBMAPTALDH1A1USP2
SCHEMBL8686162 0.89 NPC1 (0.48) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7300831 0.87 CTSS (0.44) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7300813 0.87 CTSS (0.44) TAS1R3TAS1R1HPGDPOLBMAPT
SCHEMBL7311615 0.87 ALDH1A1 (0.53) TAS1R3TAS1R1HPGDPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed