SCHEMBL7311615

SCHEMBL7311615

CCCCC(NCC(CC(C)C)NC(=O)/C=C/c1ccc(OC)cc1)C(=O)CSCc1ccco1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
MAPT P10636 5/20 0.53
HPGD P15428 3/20 0.53
TAS1R3 Q7RTX0 7/20 0.49
TAS1R1 Q7RTX1 7/20 0.49
KDM4E B2RXH2 2/20 0.42
RECQL P46063 2/20 0.39
GAA P10253 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
TDP1 Q9NUW8 2/20 0.37
HTT P42858 2/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 2/20 0.37
MEN1 O00255 1/20 0.37
GLA P06280 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7311611 0.88 TAS1R3 (0.53) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7311618 0.88 TAS1R3 (0.53) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7311608 0.88 TAS1R3 (0.53) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7300826 0.87 TAS1R3 (0.42) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7306946 0.86 ALDH1A1 (0.41) ALDH1A1MAPTHPGDRECQLGAA
SCHEMBL7306407 0.83 POLB (0.51) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7438985 0.81 ALDH1A1 (0.40) ALDH1A1MAPTHPGDKDM4ERECQL
SCHEMBL7442933 0.81 ALDH1A1 (0.44) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7311350 0.80 TAS1R3 (0.38) ALDH1A1MAPTHPGDTAS1R3TAS1R1
SCHEMBL7301797 0.80 CTSK (0.42) ALDH1A1MAPTHPGDSMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed