SCHEMBL7301411

SCHEMBL7301411

CCC1(CC)C[C]c2ccc(F)cc2O1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 11/20 0.33
HTR2C P28335 1/20 0.33
CYP3A4 P08684 1/20 0.31
KCNE1 P15382 3/20 0.30
KCNQ1 P51787 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7297848 0.88 KCNE1 (0.35) TRPV1HTR2CCYP3A4KCNE1KCNQ1
SCHEMBL7290029 0.79 AKR1B1 (0.37) TRPV1HTR2CCYP3A4
SCHEMBL7300510 0.77 CYP2D6 (0.33) CYP3A4
SCHEMBL7301405 0.71 HTR2C (0.40) TRPV1HTR2CCYP3A4KCNE1KCNQ1
SCHEMBL9983051 0.69 ADRA2A (0.38) TRPV1KCNE1KCNQ1
SCHEMBL7294345 0.69
SCHEMBL7298874 0.69 KCNE1 (0.39) CYP3A4KCNE1KCNQ1
SCHEMBL2319623 0.68 MAOB (0.47)
SCHEMBL9585171 0.67 AKR1B1 (0.39) CYP3A4
SCHEMBL3319723 0.67 TRPV1 (0.42) TRPV1HTR2CCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed