SCHEMBL7297848

SCHEMBL7297848

CCC1(CC)C[C]c2cc(F)ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 3/20 0.35
KCNQ1 P51787 3/20 0.35
TRPV1 Q8NER1 12/20 0.34
CYP3A4 P08684 1/20 0.33
AKR1B1 P15121 2/20 0.32
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301411 0.88 TRPV1 (0.33) KCNE1KCNQ1TRPV1CYP3A4HTR2C
SCHEMBL7294959 0.79 AKR1B1 (0.40) KCNE1KCNQ1TRPV1AKR1B1HTR2C
SCHEMBL7298874 0.78 KCNE1 (0.39) KCNE1KCNQ1CYP3A4
SCHEMBL7300510 0.77 CYP2D6 (0.33) CYP3A4
SCHEMBL9585171 0.76 AKR1B1 (0.39) CYP3A4AKR1B1
SCHEMBL9983051 0.72 ADRA2A (0.38) KCNE1KCNQ1TRPV1AKR1B1
SCHEMBL7297844 0.70 HTR2C (0.39) KCNE1KCNQ1TRPV1CYP3A4AKR1B1
SCHEMBL7294345 0.69
SCHEMBL7301405 0.68 HTR2C (0.40) KCNE1KCNQ1TRPV1CYP3A4AKR1B1
SCHEMBL3322611 0.68 MAPT (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5260444-A Cardiovascular, hypotensive WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-11-09 US disclosed
US-5208245-A Hypotensive agents WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1993-05-04 US disclosed
EP-0460418-A2 Novel Dihydropyridine derivative WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1991-12-11 EP disclosed