SCHEMBL7301514

SCHEMBL7301514

COc1ccc(CC(NC(=O)c2ccc(C(=N)N)cc2)C(=O)N2CCC(OC(C)=O)CC2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.62
ITGA2B P08514 8/20 0.62
CYP51A1 Q16850 1/20 0.49
KMT2A Q03164 1/20 0.49
CA2 P00918 1/20 0.47
F2 P00734 2/20 0.45
PLG P00747 2/20 0.45
F10 P00742 1/20 0.45
PLAU P00749 1/20 0.45
ST14 Q9Y5Y6 1/20 0.45
POLB P06746 1/20 0.44
CALCRL Q16602 1/20 0.44
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
TPSAB1 Q15661 1/20 0.43
TPSD1 Q9BZJ3 1/20 0.43
TPSG1 Q9NRR2 1/20 0.43
PSMB8 P28062 2/20 0.43
PSMB5 P28074 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301509 0.91 ITGB3 (0.60) ITGB3ITGA2BCYP51A1KMT2ACA2
SCHEMBL8020868 0.91 ITGB3 (0.75) ITGB3ITGA2BCYP51A1F2PLG
SCHEMBL7291927 0.89 ITGB3 (0.62) ITGB3ITGA2BCYP51A1KMT2ACA2
SCHEMBL7291943 0.89 ITGB3 (0.61) ITGB3ITGA2BCYP51A1KMT2ACA2
SCHEMBL7292028 0.87 ITGB3 (0.82) ITGB3ITGA2BCYP51A1CA2F2
SCHEMBL7284349 0.87 ITGB3 (0.82) ITGB3ITGA2BCYP51A1CA2F2
SCHEMBL9259158 0.85 ITGB3 (0.60) ITGB3ITGA2BCYP51A1KMT2ACA2
SCHEMBL8690536 0.84 ITGB3 (0.55) ITGB3ITGA2BF2PLGPOLB
SCHEMBL8689958 0.83 ITGB3 (0.73) ITGB3ITGA2BCYP51A1F2PLG
SCHEMBL27386352 0.81 ITGB3 (0.61) ITGB3ITGA2BCYP51A1CA2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0505868-B1 N-Acyl-alpha-aminoacids derivatives HOFFMANN LA ROCHE (CH) 1995-09-13 EP claimed