SCHEMBL7301945

SCHEMBL7301945

CC(C)CN(C)CCCN1CC=C(c2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.47
PPARA Q07869 2/20 0.47
PARP1 P09874 1/20 0.46
SIGMAR1 Q99720 7/20 0.42
MAPK1 P28482 1/20 0.38
HTR7 P34969 2/20 0.38
MCHR1 Q99705 1/20 0.37
DRD2 P14416 1/20 0.37
TRPV4 Q9HBA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308762 0.85 QDPR (0.48) PARP1SIGMAR1DRD2
SCHEMBL6373460 0.76 PARP1 (0.50) PPARGPPARAPARP1SIGMAR1HTR7
SCHEMBL6374865 0.72 PARP1 (0.48) PPARGPPARAPARP1SIGMAR1HTR7
SCHEMBL7104174 0.71 PARP1 (0.47) PPARGPPARAPARP1SIGMAR1DRD2
SCHEMBL16843071 0.70 SIGMAR1 (0.50) SIGMAR1DRD2
SCHEMBL11932475 0.70 SIGMAR1 (0.61) PPARGPPARAPARP1SIGMAR1HTR7
SCHEMBL8915112 0.69 QDPR (0.62) PPARGPPARA
SCHEMBL9967722 0.69 SIGMAR1 (0.56) SIGMAR1
SCHEMBL7296334 0.67 PPARG (0.56) PPARGPPARAPARP1SIGMAR1
SCHEMBL1470365 0.67 DRD4 (0.52) PARP1SIGMAR1MAPK1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149817-A Psychotropic agents SHIONOGI & CO., LTD. (JP) 1992-09-22 US disclosed
EP-0445701-A1 Novel tetrahydropyridine derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-09-11 EP disclosed