SCHEMBL7296334

SCHEMBL7296334

FC(F)(F)c1ccc(C2=CCN(CCCOc3ccc(Cl)c(Cl)c3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.56
PPARA Q07869 9/20 0.56
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TLR9 Q9NR96 1/20 0.46
SIGMAR1 Q99720 3/20 0.45
PARP1 P09874 1/20 0.44
HTR5A P47898 1/20 0.44
S1PR1 P21453 1/20 0.43
S1PR3 Q99500 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7295502 0.89 PPARG (0.63) PPARGPPARAKDM4EALDH1A1SMN1; SMN2
SCHEMBL7305418 0.86 PPARG (0.58) PPARGPPARAKDM4EALDH1A1SMN1; SMN2
SCHEMBL7529625 0.73 CARM1 (0.56) KDM4EALDH1A1SMN1; SMN2
SCHEMBL6373460 0.72 PARP1 (0.50) PPARGPPARASIGMAR1PARP1
SCHEMBL6374865 0.71 PARP1 (0.48) PPARGPPARASIGMAR1PARP1
SCHEMBL7230184 0.70 MAOA (0.62) KDM4EALDH1A1SMN1; SMN2HTR5A
SCHEMBL7564110 0.70 KDM4E (0.82) KDM4EALDH1A1SMN1; SMN2
SCHEMBL7104174 0.69 PARP1 (0.47) PPARGPPARASIGMAR1PARP1
SCHEMBL4589510 0.69 PPARG (0.64) PPARGPPARAS1PR1S1PR3
SCHEMBL2928576 0.68 HTR6 (0.44) PPARGPPARASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5149817-A Psychotropic agents SHIONOGI & CO., LTD. (JP) 1992-09-22 US disclosed
EP-0445701-A1 Novel tetrahydropyridine derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-09-11 EP disclosed