SCHEMBL7302599

SCHEMBL7302599

O=Cc1cccc2oc(-c3ccccc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.47
RCE1 Q9Y256 1/20 0.43
RAB9A P51151 7/20 0.42
SMN1; SMN2 Q16637 7/20 0.42
HIF1A Q16665 1/20 0.42
HTR3A P46098 1/20 0.41
NPC1 O15118 6/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CASP3 P42574 3/20 0.40
SENP7 Q9BQF6 3/20 0.40
SENP6 Q9GZR1 3/20 0.40
SENP8 Q96LD8 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
POLB P06746 1/20 0.40
ELANE P08246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4583536 0.86 HTR3A (0.44) TOP2ASMN1; SMN2HTR3AMEN1KMT2A
SCHEMBL6045554 0.83 ERN1 (0.49) TOP2ARAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL2109256 0.77 ERN1 (0.53) TOP2ARAB9ASMN1; SMN2NPC1MEN1
SCHEMBL1618212 0.76 TOP2A (0.58) TOP2ARCE1RAB9ASMN1; SMN2HIF1A
SCHEMBL11561655 0.76 NPC1 (0.45) TOP2ARAB9ASMN1; SMN2NPC1MEN1
SCHEMBL121325 0.75 TOP2A (0.65) TOP2ARCE1RAB9ASMN1; SMN2HIF1A
SCHEMBL6297297 0.75 ELANE (0.45) MEN1KMT2AALDH1A1MAPTL3MBTL1
SCHEMBL7109574 0.75 RAB9A (0.53) TOP2ARCE1RAB9ASMN1; SMN2HIF1A
SCHEMBL22085386 0.75 SMN1; SMN2 (0.56) TOP2ARCE1RAB9ASMN1; SMN2HIF1A
SCHEMBL56593 0.75 TOP2A (0.53) TOP2ARCE1RAB9ASMN1; SMN2HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5412099-A Intermediate benzothiazolyl- and benzoxazolyl-aldehyde compounds BAYER AKTIENGESELLSCHAFT (DE) 1995-05-02 US disclosed
EP-0450420-B1 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1994-09-21 EP disclosed
US-5254692-A Inotropic BAYER AKTIENGESELLSCHAFT (DE) 1993-10-19 US disclosed
US-5200420-A Inotropic agents for cardiovascular disorders BAYER AKTIENGESELLSCHAFT (DE) 1993-04-06 US disclosed
EP-0450420-A2 Dihydropyridines substituted by heterocycles, process for their preparation and their use in medicaments BAYER AG (DE) 1991-10-09 EP disclosed